Tadalafil hmoov (CAS 171596-29{23}}5), tshuaj hu ua (6R,12aR)-6-(1,3-benzodioxol-5-yl)-2-methyl-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[3,4-b]indole-dawb hmoov, tsis muaj ntxhiab-1,4 thiab me ntsis soluble hauv dej, yooj yim soluble hauv dimethyl sulfoxide (DMSO) thiab ethanol. Nws yog ib qho tseem ceeb raw khoom nyob rau hauv high-end txiv neej noj qab haus huv cov tshuaj, lug siv nyob rau hauv zus tau tej cov tshuaj ntsiav, ntsiav tshuaj, thiab cov kua qhov ncauj. Tadalafil yog ib qho kev xaiv inhibitor ntawm phosphodiesterase type 5 (PDE5), uas ua haujlwm los ntawm inhibiting degradation ntawm cyclic guanosine monophosphate (cGMP) nyob rau hauv cov leeg nqaij, so cov leeg du ntawm lub corpus cavernosum, txhawb cov ntshav txaus, thiab pab txhim kho txiv neej kev ua haujlwm. Piv nrog Sildenafil, Tadalafil muaj ib nrab-lub neej ntev (txog 36 teev), uas txhais tau hais tias nws tuaj yeem muab cov nyhuv ntev dua, tso cai rau cov neeg siv sijhawm siv tau yooj yim dua, thiab muaj kev phiv tsawg dua, ua rau nws nrov ntawm cov neeg siv khoom.
Peb Tadalafil bulk hmoov yog tsim los ntawm advanced synthesis technology thiab nruj zoo tswj txheej txheem, kom ntseeg tau tias txhua batch ntawm cov khoom muaj siab purity, ruaj khov zoo, thiab tsis muaj teeb meem impurities. Cov khoom lag luam muaj cov ntsiab lus tsis tshua muaj hlau hnyav (tsawg dua lossis sib npaug li 5ppm), ua tau raws li cov qauv kev lag luam thoob ntiaj teb, thiab tsim nyog rau ntau yam siab - kawg txiv neej kev noj qab haus huv formulations. Nws tuaj yeem siv ib leeg lossis sib xyaw nrog lwm cov khoom siv raw xws li Sildenafil thiab Vardenafil los txhim kho cov nyhuv thiab ua tau raws li cov kev xav tau ntawm cov neeg siv khoom sib txawv. Nrog rau kev txhim kho txuas ntxiv ntawm cov txiv neej cov khoom lag luam kev noj qab haus huv, qhov kev thov rau Tadalafil raw khoom yog nce xyoo los ntawm lub xyoo, thiab peb cov khoom tuaj yeem muab rau koj nrog siab -zoo, nqi- cov kev daws teeb meem zoo los pab koj kom tau txais txiaj ntsig zoo hauv kev lag luam siab - kawg.
Specification & Parameters
|
Lub npe Parameter |
Specification |
Txoj Kev Xeem |
|
CAS Nr |
171596-29-5 |
HPLC |
|
Molecular Formula |
C22H19N3O4 |
Elemental Analysis |
|
Molecular Luj |
389.40 |
Kev suav Molecular Luj |
|
Purity |
Ntau dua lossis sib npaug li 99.5% |
HPLC |
|
Qhov tshwm sim |
Dawb rau tawm -dawb crystalline hmoov |
Kev tshuaj xyuas qhov muag |
|
Melting Point |
298-302 degree |
Melting Point Tester |
|
Poob rau ziab |
Tsawg dua lossis sib npaug li 0.3% |
105 degree, 2 h |
|
Cov ntsiab lus hnyav hlau |
Tsawg dua lossis sib npaug li 5ppm |
Atomic Absorption Spectrometry |
|
Residue ntawm Ignition |
Tsawg dua lossis sib npaug li 0.1% |
Ignition Method |
|
Solubility |
Me ntsis soluble hauv dej, soluble hauv DMSO thiab ethanol |
Solubility Test |
|
Ib nrab -Lub neej |
Mus txog 36 teev |
Pharmacokinetic Test |
|
Kev cia khoom |
Khaws rau hauv qhov chaw txias, qhuav, thiab zoo- qhov cua, deb ntawm lub teeb thiab noo noo, ntawm 2-8 degree |
Kev kuaj cia |
|
Txee lub neej |
24 lub hlis (nyob rau hauv kev cia zoo) |
Kev kuaj kev ruaj ntseg |
Qhov Zoo & Nta
Ntev -Kev Ua Haujlwm Zoo: Nrog ib nrab ntawm - lub neej ntev txog 36 teev, nws muab cov txiaj ntsig ntev dua - ntev dua li lwm cov khoom siv raw zoo sib xws (xws li Sildenafil), ua rau cov neeg siv sijhawm siv tau yooj yim dua, txhim kho cov neeg siv kev paub thiab cov khoom sib tw.
High Purity & Kev Nyab Xeeb: Purity Ntau dua los yog sib npaug rau 99.5%, tsis muaj teeb meem impurities, cov ntsiab lus hlau hnyav tsawg dua lossis sib npaug li 5ppm, raws li cov qauv kev lag luam thoob ntiaj teb. Kev tswj hwm nruj nruj los ntawm kev xaiv cov khoom siv raw rau kev tsim khoom, ua kom cov khoom muaj kev nyab xeeb thiab ua haujlwm zoo, txo qhov kev pheej hmoo ntawm kev phiv.
Kev ruaj ntseg zoo & khoom siv: Txais siv thev naus laus zis synthesis thiab automated ntau lawm kab, cov khoom zoo yog ruaj khov, thiab batch -rau -batch sib txawv me me. Peb muaj cov zis txhua hli ntawm 4000kg, uas tuaj yeem ua tau raws li cov kev xav tau ntawm cov neeg siv khoom ntau thiab xyuas kom meej ntawm - lub sijhawm xa khoom.
Tus nqi sib tw: Lub Hoobkas- muag ncaj qha, tsis muaj neeg nruab nrab, ncaj qha txo tus nqi yuav khoom rau cov neeg siv khoom. Peb muab tus nqi hloov pauv raws li qhov kev txiav txim kom muaj nuj nqis, thiab muab cov luv nqi ntxiv rau cov neeg siv khoom sib koom ua ke ntev -.
Ua tiav Daim Ntawv Pov Thawj & Ua Raws Cai: Tau nruab nrog ISO9001, GMP, COA, MSDS, thiab thib peb- cov ntaub ntawv kuaj xyuas tog neeg (SGS, Intertek), ua raws li EU, US, thiab thoob ntiaj teb cov cai tswj kev lag luam, pab cov neeg siv khoom sai dhau kev lis kev cai thiab kev tshuaj xyuas kev lag luam.
Yooj yim rau Formula: Cov khoom yog cov hmoov dawb crystalline hmoov nrog zoo solubility thiab ruaj khov, yooj yim rau kev sib xyaw nrog lwm cov ntaub ntawv raw, haum rau ntau yam txheej txheem xws li tshuaj ntsiav, ntsiav tshuaj, thiab cov kua hauv qhov ncauj, txo qhov nyuaj ntawm kev tsim khoom.
Tsawg Qhov Teeb Meem: Piv nrog rau lwm cov khoom siv raw zoo sib xws, peb cov hmoov Tadalafil bulk muaj kev phiv tsawg dua, xws li mob taub hau, yaug, thiab kiv taub hau, ua rau nws nrov dua ntawm cov neeg siv khoom thiab txhim kho kev lag luam kev lees paub ntawm cov khoom kawg.
Lub zog & muaj peev xwm
Peb yog cov chaw tsim khoom ntawm cov khoom siv tshuaj thiab kev noj qab haus huv nrog 10+ xyoo ntawm kev paub hauv R&D, ntau lawm, thiab xa tawm. Peb lub hauv paus tsim khoom yog nyob rau hauv high-tech industrial park, npog thaj tsam ntawm 20,000 square metres, nruab nrog cov khoom siv ntau lawm thiab cov cuab yeej ntsuas, suav nrog HPLC, GC, atomic absorption spectrometer, thiab cov khoom siv tshuaj pharmacokinetic, kom ntseeg tau tias txhua pawg ntawm cov khoom ua tau raws li cov qauv zoo tshaj plaws. Peb muaj cov kws tshaj lij R & D pab pawg tsim los ntawm 15+ cov kws tshaj lij engineers thiab cov kws tshaj lij, uas tau cog lus rau cov khoom lag luam thiab kev txhim kho kom zoo, thiab tuaj yeem muab kev txhawb nqa thiab kev daws teeb meem rau cov neeg siv khoom.
Peb cov khoom lag luam txhua xyoo ntawm Tadalafil bulk hmoov nce mus txog 48,000kg, nrog rau kev ua tiav cov saw hlau, los ntawm cov khoom siv raw khoom mus rau cov khoom xa tuaj, tsim ib qho kev pabcuam nres. Peb tau txais ISO9001 cov ntawv pov thawj kev tswj hwm zoo thiab GMP daim ntawv pov thawj, thiab peb cov khoom raug xa tawm mus rau ntau tshaj 60 lub teb chaws thiab cheeb tsam, suav nrog Tebchaws Meskas, Europe, Southeast Asia, thiab Middle East, thiab tau tsim ntev -kev sib raug zoo nrog ntau yam zoo- paub txog cov tuam txhab khoom noj qab haus huv thiab cov chaw tsim tshuaj. Peb muaj pab pawg muag khoom tshaj lij thiab tom qab- pab pawg muag khoom, muab kev sib tham hauv online 24/7 thiab tom qab{12}} kev muag khoom, daws txhua qhov kev yuav khoom thiab siv cov teeb meem rau cov neeg siv khoom raws sijhawm.
Tsis tas li ntawd, peb muab qhov tseem ceeb rau kev tiv thaiv ib puag ncig thiab kev txhim kho kom ruaj khov, siv cov thev naus laus zis ntsuab, txo cov pa phem ib puag ncig, thiab ua raws li cov qauv kev tiv thaiv thoob ntiaj teb. Peb cov txheej txheem tsim khoom tau dhau qhov kev tshuaj xyuas ib puag ncig, kom ntseeg tau tias cov txheej txheem tsim khoom yog ib puag ncig tus phooj ywg thiab ruaj khov.

